Raloxifene For Gyno: Is It The Best SERM PCT For Stopping The Moobs?
I’m going to talk to you about raloxifene. I’ll tell you what it’s used for, and also why loads of men are now using it to treat the symptoms of gyno.
Don’t worry, we will go slow and simple here, but give you enough information to make a great decision on whether raloxifene is the best choice for you in terms of countering problems with low testosterone and elevated estrogen, especially in comparison to Tamoxifen (Nolvadex) and Clomid (Clomiphene Citrate).
We will cover the basics around what causes gyno, through to giving you a comparison between the three main SERMs (Selective Estrogen Receptor Modulators) out there that you can use to counter it both on cycle.
I’ll also explain how SERMs are different to aromatase inhibitors (AIs) and why it’s absolutely crucial that you don’t get the two different types of estrogen regulating chemicals confused.
Plus, I’ll tell you exactly how to use it, and for how long. As well as all that, and also conclude by telling you where you can actually find raloxifene for sale that is trustworthy.
Let’s Talk About Gyno
I think we should start by saying exactly what gyno is. It’s a slang term for something called Gynecomastia. That’s the official medical term to describe male breast tissue growth.
Although it can happen to men any stage of their lives naturally, it can be brought on when using androgenic SARMs. Selective androgen receptor modulators which mimic testosterone. I’ll cover exactly how they can cause gyno in detail in a moment.
You can spot gyno amongst a range of other symptoms brought on by excess estrogen. You may notice feminine things happening, but it’s a puffiness around your nipples that is the dead giveaway. It feels like excess fat, but it’s not.
Alongside this production of tissue on the male breast, you can get decrease in male muscle tissue in the breast area as well. Put together, you got a real problem.
Gyno is difficult to reverse once it stops, but raloxifene appears to be one of the few ways that you potentially can without surgery.
What Causes Gyno & Can You Avoid It With PCT?
What actually causes gyno is an excess of estrogen. This is usually coupled with a decrease in testosterone.
What happens is testosterone is converted into estrogen which exacerbates a problem which may already be there.
Using SARMs can make things far worse. SARMs convince your body that they have higher levels of testosterone present than there are in reality.
So your body reacts as if it’s got high levels of testosterone, which is brilliant for muscle building, and all the things you associate with high levels of testosterone.
However, your body is panicking because you’ve got these elevated levels of testosterone, so it cuts its own production levels. So even though you feel fantastic, your testosterone is dropping through the floor. Your body is being fooled and so are you.
This leads to an imbalance where the estrogen in your body is too high in comparison, and can be made worse when it eats up more testosterone. Testosterone gets converted into estrogen, and the more estrogen there is then the higher this conversion would be.
Can you avoid it were PCT? The simple answer is yes.
These are the options you have for PCT to try and avoid gyno:
- 1. Keep your androgenic SARMs cycles a short as possible. Immediately at the end of the cycle use Nolvadex, or Clomid if you feel a real testosterone drop, at high doses, tapering down after a couple of weeks.
- 2. If you don’t want to cut your cycle short and you can feel the effects of low testosterone, then you can use Nolvadex on cycle to try and counter it. I wouldn’t recommend this though because you are exacerbating the problem.
- 3. Your third option is to cut the SARMs cycle short. Immediately start Nolvadex treatment, if it’s a real feeling your T levels drop through the floor, then use the far stronger Clomid.
Your Options When You Suspect You Have Gyno
You’ll have noticed I haven’t mentioned raloxifene as a PCT supplement. I’ve only talked about Nolvadex and Clomid.
I’ll discuss it in more detail in a little while, but basically raloxifene has been found in studies to be better for dealing with gyno symptoms, but less effective for allowing testosterone to bounce back. That may sound counterintuitive, and we will go into detail in a little while.
So if you suspect you have gyno, you have the following options, both in terms of self-medication, and seeking help:
- Androgen therapy
- DHT therapy
- Anti-estrogen therapy
Some of those are quite invasive, and I’m hoping you would allow things to get that far in terms of breast tissue development and the effects of estrogen ravaging your male body before you took action.
So we are looking at heading off with Nolvadex or Clomid, or intervening more heavily and efficiently with relax is seen either as a preventative measure, or to deal with physical symptoms.
What Is Raloxifene?
Raloxifene is classed as a SERM – a Selective Estrogen Receptor Modulator. This is also the case with tamoxifen (Nolvadex) and Clomid.
They all work in the same way, by binding to estrogen receptors, thus blocking them from being blinded to buy estrogen itself. They therefore halt the mechanism of estrogen in the body, but don’t stop its production.
Another class of drugs which people get confused with our aromatase inhibitors, of which the best known example is letrozole.
Aromatase inhibitors work by blocking the action of aromatase, which is crucial to the production of estrogen. So in aromatase inhibitor blocks the production of estrogen, rather than just blocking its binding to estrogen receptors.
So raloxifene is basically the same as Nolvadex and Clomid, so what makes it better for gyno?
The bottom line is that studies have shown that raloxifene is better at inhibiting estrogen receptor action in breast tissue than Nolvadex or Clomid.
Don’t ask me why, I don’t understand science, and the studies I’ve read don’t make it clear. But they all conclude the same thing: raloxifene works better for stopping and reducing gyno than any other SERM.
How To Use Raloxifene For Bodybuilding Gyno Symptoms
So that’s the background to why people advocate using raloxifene for bodybuilding gyno, but how do you actually use it?
Use of raloxifene will lower circulating estrogen levels significantly. Now you don’t want to do this for long, because low estrogen can actually cause problems in men as well. Men seem to be all about testosterone, but low estrogen can affect bone density.
Raloxifene has about 10 times the power binding affinity to the estrogen receptors in male breast tissue than other SERM PCT supplements.
If you suspect you’ve got gyno, or you want to head it off because you’re concerned, then hit yourself with raloxifene at the beginning of your PCT cycle.
You could use it alongside tamoxifen or clomiphene, but make sure you watch your overall dosage isn’t too high.
You can even use the locks 15 on cycle, meaning you can carry on your SARMs cycle while targeting the growing levels of estrogen and stopping them binding to breast tissue is easily.
I wouldn’t really recommend that, and when you feel T level drops, or you suspect dynamite kicking, stop the cycle and focus on reversal.
Here’s how to use raloxifene:
- You’ll want to dose it at around 60 mg per day. Slightly lower if you’re going to run it with Nolvadex.
- Use raloxifene if you suspect you are at risk of gyno, or if you actually can feel excess breast tissue (lumps in the breast that weren’t there before).
- It’s possible that the locks of theme can actually diminish this excess breast tissue. But that will take a few weeks of using it.
- Make sure your raloxifene dosage is around 60 mg for the first two weeks, and then taper it down to around half that over the next two weeks.
- Nolvadex is well tolerated and has been proven to shrink gyno as well. If the raloxifene isn’t doing it on its own, then consider stacking it so that you can try and attack the breast tissue problem better.
I’ll just finish this section by saying I wouldn’t advise you stack raloxifene with an aromatase inhibitor. In fact, I don’t really suggest you use an aromatase inhibitor at all.
SERMs allow your testosterone levels to bounce back, whereas aromatase inhibitors stop the production.
So you’ll get higher levels of testosterone, and your estrogen levels will drop dramatically. However, what most guys don’t realize is that this can lead to brittle bones. If you keep using aromatase inhibitors to bounce your testosterone levels back, you could be storing up some significant bone health problems for the future.
Is Raloxifene For Men Safe?
Raloxifene at sensible doses for short duration seems to be perfectly safe. It’s a SERM, and people have been using Nolvadex and Clomid for two decades after SARMs and steroid cycles without issues.
That doesn’t mean it’s not without side effects though. These are the sort of raloxifene side effects you should watch out for:
- Joint pain
- Hot flushes
- Muscle or bone weakness
Overall, at doses of 60 mg or less, taken for no more than 4-8 weeks, you should be fine. But you need to be in tune with your body to ensure that you are not creating bigger problems than you are trying to solve.
Raloxifene Review Conclusion
So the conclusion of my raloxifene gyno guide is that it’s a superior SERM if you want to deal specifically with gyno symptoms.
Because it combines with a higher affinity to estrogen receptors in breast tissue it better at stopping the growth of breast tissue than any other drugs in the same class.
But I will say as part of the conclusion to this review of raloxifene that it’s far better to never get to the stage where you have excess breast tissue to worry about in the first place.
I’ve never suffered from gyno, but a friend of mine has. It wasn’t pleasant, and he was an idiot.
If unfortunately you have already got the stage where you can feel small lumps of excess tissue, and I’m telling you that raloxifene is your best hope. Hit yourself with 60 mg right now, and maybe pair it up with Nolvadex after a few weeks if it’s not working. That’s your best bet, before you have to look at surgical intervention.
Finding Raloxifene For Sale
Let me finish here then by telling you where you can actually find raloxifen for sale.
As with all bodybuilding supplements it’s a grey market product. It was never designed for men, and certainly not for bodybuilders, so it’s never going to be prescribed, or even available off label.
But you can buy on the grey market in generic form. Reconstructed for sale without prescription or oversight.
The best place I found to buy raloxifene is Swiss Chems. They sold me high-quality SARMs and supplements for three years now and I haven’t ever had a problem.
Raloxifene costs $85.95 from Swiss Chems. For your money you’ll get 60 capsules, each dosing 20 mg.
Start with three capsules per day (total dose 60 mg) and see how you feel after two weeks. Then drop down to 40 mg, and see how that goes.
If after a month you not seeing a reversal, then you can either up the dose again, preferably, pair it up with 30 mg or so of Nolvadex.
I wouldn’t suggest you persist with this level of PCT for more than two months though, because of how it can impact the balance between estrogen and testosterone causing further problems.